RT Book, Section A1 Rollins, Douglas E. A1 Blumenthal, Donald K. SR Print(0) ID 1140226452 T1 Cancer Chemotherapy and Cytotoxic Agents T2 Workbook and Casebook for Goodman and Gilman's The Pharmacological Basis of Therapeutics YR 2016 FD 2016 PB McGraw-Hill Education PP New York, NY SN 9780071793360-qa LK accesspharmacy.mhmedical.com/content.aspx?aid=1140226452 RD 2024/04/18 AB Table Graphic Jump Location|Download (.pdf)|PrintTable 45-3. AntimetabolitesTYPE OF AGENTNONPROPRIETARY NAMESDISEASEFolic acid analogsMethotrexate (amethopterin)Acute lymphocytic leukemia; choriocarcinoma; breast, head, neck and lung cancers; osteogenic sarcoma; bladder cancerPemetrexedMesothelioma, lung cancerPyrimidine analogsFluorouracil (5-fluorouracil; 5-FU), capecitabineBreast, colon, esophageal, stomach, pancreas, head and neck; premalignant skin lesion (topical)Cytarabine (cytosine arabinoside)Acute myelogenous and acute lymphocytic leukemia; non-Hodgkin’s lymphomaGemcitabinePancreatic, ovarian, lung cancer5-aza-cytidineMyelodysplasiaDeoxy-5-aza-cytidineMyelodysplasiaPurine analogs and related inhibitorsMercaptopurine (6-mercaptopurine; 6-MP)Acute lymphocytic and myelogenous leukemia; small cell non-Hodgkin’s lymphomaPentostatin (2’-deoxycoformycin)Hairy cell leukemia; chronic lymphocytic leukemia; small cell non-Hodgkin’s lymphomaFludarabineChronic lymphocytic leukemiaClofarabineAcute myelogenous leukemiaNelarabineT-cell leukemia, lymphoma